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Tranexamic Acid

Medically reviewed: Dr. Murat Toktamışoğlu · 2026-05-21

Definition

Hemostatic agent; oral 250 mg 2x/day or topical 3-5% — recent star in melasma treatment.

Detail

Inhibits melanocyte-to-keratinocyte melanin transfer. Adjunct for stubborn melasma. Contraindicated: thrombosis history, hormonal medication + smoking.

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